An intranasal nanoparticle STING agonist protects against respiratory viruses in animal models.

Publication date: Jul 18, 2024

Respiratory viral infections cause morbidity and mortality worldwide. Despite the success of vaccines, vaccination efficacy is weakened by the rapid emergence of viral variants with immunoevasive properties. The development of an off-the-shelf, effective, and safe therapy against respiratory viral infections is thus desirable. Here, we develop NanoSTING, a nanoparticle formulation of the endogenous STING agonist, 2′-3′ cGAMP, to function as an immune activator and demonstrate its safety in mice and rats. A single intranasal dose of NanoSTING protects against pathogenic strains of SARS-CoV-2 (alpha and delta VOC) in hamsters. In transmission experiments, NanoSTING reduces the transmission of SARS-CoV-2 Omicron VOC to nacEFve hamsters. NanoSTING also protects against oseltamivir-sensitive and oseltamivir-resistant strains of influenza in mice. Mechanistically, NanoSTING upregulates locoregional interferon-dependent and interferon-independent pathways in mice, hamsters, as well as non-human primates. Our results thus implicate NanoSTING as a broad-spectrum immune activator for controlling respiratory virus infection.

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Concepts Keywords
Mice Administration, Intranasal
Nanoparticle Animals
Therapy Antiviral Agents
Vaccination Antiviral Agents
Viruses COVID-19
Cricetinae
Disease Models, Animal
Female
Humans
Male
Membrane Proteins
Membrane Proteins
Mice
Nanoparticles
Nucleotides, Cyclic
Nucleotides, Cyclic
Orthomyxoviridae Infections
Rats
SARS-CoV-2
Sting1 protein, mouse

Semantics

Type Source Name
disease VO Viruses
disease MESH viral infections
disease MESH morbidity
drug DRUGBANK Spinosad
disease VO vaccination
disease VO effective
disease VO dose
drug DRUGBANK Oseltamivir
disease MESH influenza
disease VO Primates
drug DRUGBANK Vinorelbine
disease MESH severe acute respiratory syndrome
disease MESH Middle East respiratory syndrome
drug DRUGBANK Esomeprazole
disease VO Optaflu
disease VO Respiratory syncytial virus
disease MESH COVID 19 pandemic
disease IDO emerging pathogen
disease MESH mutation rate
disease VO ineffective
disease IDO replication
disease MESH infection
disease IDO host
disease IDO innate immune response
pathway REACTOME Immune System
disease VO USA
disease MESH asymptomatic infection
disease MESH defects
drug DRUGBANK Isoxaflutole
drug DRUGBANK Guanosine
drug DRUGBANK Phosphate ion
disease MESH reinfection
disease VO viability
disease VO dead
disease VO time
disease MESH inflammation
disease IDO blood
disease IDO cell
disease VO frequency
disease VO volume
disease VO efficient
disease VO stomach
drug DRUGBANK Coenzyme M
disease MESH body weight changes
disease MESH weight loss
disease IDO process
drug DRUGBANK Cyclic Guanosine Monophosphate
drug DRUGBANK Adenosine phosphate
disease MESH Disease Models Animal
disease MESH Orthomyxoviridae Infections

Original Article

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